Carbetocin , 98％
Synonym(s):
N-(4-Mercapto-1-oxobutyl)-O-methyl-L-tyrosyl-L-isoleucyl-L-glutaminyl-L-asparaginyl-L-cysteinyl-L-prolyl-L-leucyl-glycinamidecyclic (1-5)-thioether acetate
CAS NO.：
Empirical Formula: C45H69N11O12S
Molecular Weight: 988.17
MDL number: MFCD01076600
EINECS: 253-312-6
| Pack Size | Price | Stock | Quantity |
| 5mg | RMB359.20 | In Stock |
|
| 10mg | RMB639.20 | In Stock |
|
| 50mg | RMB2399.20 | In Stock |
|
| 100mg | RMB4639.20 | In Stock |
|
| others | Enquire |
PRODUCT Properties
| Melting point: | 140 - 160°C |
| Boiling point: | 1477.9±65.0 °C(Predicted) |
| alpha | D -69.0° (c = 0.25 in 1M acetic acid) |
| Density | 1.218±0.06 g/cm3(Predicted) |
| storage temp. | -15°C |
| solubility | DMSO (Slightly), Methanol (Slightly) |
| form | powder |
| pka | 13.07±0.70(Predicted) |
| color | white to beige |
| Water Solubility | Soluble to 29.65 mg/ml in water |
| Stability: | Hygroscopic |
| InChIKey | NSTRIRCPWQHTIA-FOILTOEQNA-N |
Description and Uses
Carbetocin is an alternative synthetic oxytocin-receptor agonist available in Canada, the United Kingdom, and other countries，but not the United States. A large multinational randomized noninferiority trial (N=29,645) found that carbetocin was noninferior to oxytocin for prevention of postpartum hemorrhage and need for additional uterotonic agents after vaginal delivery. Carbetocin has a longer duration of action than oxytocin, eliminating the need for prolonged infusion.
Carbetocin is an obstetric drug used to control postpartum hemorrhaging.
A new synthetic analog of oxytocin, carbetocin, is long acting and also has a rapid onset of action. It is an oxytocin receptor agonist and also stimulates milk let down due to its action on oxytocin receptors of myoepithelial cells.
