M6080335
Tianeptine , BR , 72797-41-2
CAS NO.：72797-41-2
Empirical Formula: C21H25ClN2O4S
Molecular Weight: 436.95
MDL number: MFCD00865376
EINECS: 276-851-9
| Pack Size | Price | Stock | Quantity |
| 5mg | RMB467.20 | In Stock |
|
| 25mg | RMB1635.20 | In Stock |
|
| others | Enquire |
Update time: 2022-07-08
PRODUCT Properties
| Melting point: | 129-131?C |
| Boiling point: | 609.2±65.0 °C(Predicted) |
| Density | 1.38±0.1 g/cm3(Predicted) |
| vapor pressure | 0.001Pa at 25℃ |
| storage temp. | Refrigerator, Under Inert Atmosphere |
| pka | 4.75±0.10(Predicted) |
| form | solid |
| InChIKey | JICJBGPOMZQUBB-UHFFFAOYSA-N |
| SMILES | C(O)(=O)CCCCCCNC1C2=CC=C(Cl)C=C2S(=O)(=O)N(C)C2=CC=CC=C21 |
| LogP | 2.162 at 25℃ and pH6 |
Description and Uses
Tricyclic compound with psychostimulant, anti-ulcer and anti-emetic properties. It is used mainly in the treatment of major depressive disorder and may also be used to treat anxiety, asthma, and irritable bowel syndrome. It has been found to act as an atypical agonist of the μ-opioid receptor with clinically negligible effects on the δ- and κ-opioid receptors. Tianeptine prevents chronic stress-induced morphological changes in the hippocampus and amygdala and blocks the effects of acute stress on synaptic plasticity in the hippocampus and PFC.
Safety
| Symbol(GHS) |  GHS08 |
| Signal word | Warning |
| Hazard statements | H362-H361-H373 |
| Precautionary statements | P201-P260-P263-P264-P270-P308+P313-P260-P314-P501-P201-P202-P281-P308+P313-P405-P501 |
| WGK Germany | 3 |
