S8937514
≥98%(HPLC),powder , 35873-49-5
Synonym(s):
8-Cyclopentyltheophylline;CPT
Pack Size | Price | Stock | Quantity |
100mg | RMB1951.58 | In Stock |
|
others | Enquire |
Update time: 2022-07-08
PRODUCT Properties
Melting point: | 250-252°C |
Boiling point: | 513.1±42.0 °C(Predicted) |
Density | 1.332±0.06 g/cm3(Predicted) |
storage temp. | -20°C Freezer |
solubility | H2O: <0.28 mg/mL, slightly soluble |
form | crystalline |
pka | 8.91±0.70(Predicted) |
color | white or off-white |
Water Solubility | Soluble in 0.1M NaOH. Slightly soluble in water. Also soluble in DMSO at 16mg/ml at 60°C. |
Stability: | Store in freezer; Solutions at 4 deg C stable for several days |
Description and Uses
A selective A1 adenosine receptor antagonist. Binding activity in rat brain membranes: Ki = 10.9 nM (A1 receptor); Ki = 1440 nM (A2 receptor).
Safety
WGK Germany | 3 |
RTECS | XH5093600 |
HS Code | 29339900 |
Toxicity | mouse,LD50,intraperitoneal,200mg/kg (200mg/kg),Journal of Medicinal Chemistry. Vol. 14, Pg. 1202, 1971. |