Pazinaclone , 0.99 , 103255-66-9

CAS NO.：103255-66-9

Empirical Formula: C25H23ClN4O4

Molecular Weight: 478.93

MDL number: MFCD00864702

PRODUCT Properties

• Melting point: 238-239°
• Boiling point: 712.5±60.0 °C(Predicted)
• Density: 1.48±0.1 g/cm3(Predicted)
• pka: 1.62±0.30(Predicted)

Description and Uses

Pazinaclone is a nonbenzodiazepine partial agonist. Animal work has shown that it has anxiolytic and anticonvulsant activity. Pazinaclone does not, however, produce the sedative, muscle relaxant, or motor coordination effects seen with diazepam (Waka and Fukada 1991). Phase II clinical trials are currently under way in the United States, Europe, and Japan, which have so far demonstrated that it is well tolerated and seems to cause significantly less sedation than do benzodiazepines (Uchiumi et al. 1992).

Anti-anxiety agent.