(1R,3S,4S)-2-(tert-Butoxycarbonyl)-2-azabicyclo[2.2.1]heptane-3-carboxylic acid , 97% , 291775-59-2

CAS NO.：291775-59-2

Empirical Formula: C12H19NO4

Molecular Weight: 241.28

MDL number: MFCD11099876

Pack Size	Price	Stock	Quantity
1g	RMB214.40	In Stock
5g	RMB661.60	In Stock
10g	RMB1150.40	In Stock
25g	RMB2061.60	In Stock
100g	RMB6206.40	In Stock
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Update time: 2022-07-08

PRODUCT Properties

Melting point:	147-152 °C
Boiling point:	371.0±25.0 °C(Predicted)
Density	1.232±0.06 g/cm3(Predicted)
storage temp.	Sealed in dry,Room Temperature
pka	4.05±0.20(Predicted)
optical activity	[α]22/D -170±10°, c = 1 in chloroform
InChIKey	IFAMSTPTNRJBRG-YIZRAAEISA-N

Description and Uses

(1R,3S,4S)-2-(tert-Butoxycarbonyl)-2-azabicyclo[2.2.1]heptane-3-carboxylic Acid is a building block in the synthesis of Ledipasvir, a potent, once-??daily oral NS5A inhibitor for the treatment of Hepatitis C Virus infection. It is also used to prepare potent direct inhibitors of factor Xa which carries significant promise for developing effective and safe anticoagulants.

Safety

Symbol(GHS)	GHS07,GHS08,GHS09
Signal word	Danger
Hazard statements	H315-H319-H335-H360-H400
Precautionary statements	P201-P273-P302+P352-P305+P351+P338-P308+P313
Hazard Codes	Xi,N
Risk Statements	61-36/37/38
Safety Statements	53-26-61
RIDADR	UN 3077 9/PG 3
WGK Germany	3

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