Mrs1706 , 98% , 264622-53-9

Synonym(s):
8-[4-[((4-Acetylphenyl)carbamoylmethyl)oxy]phenyl]-1,3-di(n-propyl)xanthine;MRS 1706;MRS1706;N-(4-Acetylphenyl)-2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)phenoxy)acetamide;N-(4-Acetylphenyl)-2-[4-(2,3,6,9-tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl)phenoxy]acetamide

CAS NO.：264622-53-9

Empirical Formula: C27H29N5O5

Molecular Weight: 503.55

MDL number: MFCD06798374

PRODUCT Properties

• Density: 1.293±0.06 g/cm3(Predicted)
• storage temp.: Sealed in dry,2-8°C
• solubility: DMSO : 6.4 mg/mL (12.71 mM; Need ultrasonic and warming)H2O : < 0.1 mg/mL (insoluble)
• form: Powder
• pka: 8.25±0.70(Predicted)
• color: Off-white to yellow

Description and Uses

MRS1706 is a selective adenosine A_2B receptor inverse agonist with K_i values of 1.39, 157, 112, and 230 nM for human A_2B, A₁, A_2A, and A₃ receptors, respectively.

MRS 1706 is a selective and potent Adenosine A2B-R inverse agonist Ki (binding affinity) values of 1.39, 157, 112, and 230 nM for human A2B, A1, A2A, and A3 receptors, respectively.