BD0553853
(R)-N-((R)-1-(4-((1H-1,2,4-Triazol-1-yl)methyl)-4-cyclohexylpiperidin-1-yl)-3-(4-chlorophenyl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide , 98% , 312637-48-2
CAS NO.：312637-48-2
Empirical Formula: C33H41ClN6O2
Molecular Weight: 589.17
MDL number: MFCD09970598
| Pack Size | Price | Stock | Quantity |
| 10mg | RMB742.40 | In Stock |
|
| 25mg | RMB1261.60 | In Stock |
|
| 50mg | RMB2018.40 | In Stock |
|
| 100mg | RMB3228.80 | In Stock |
|
| others | Enquire |
Update time: 2022-07-08
PRODUCT Properties
| Density | 1.33±0.1 g/cm3(Predicted) |
| storage temp. | Store at -20°C |
| solubility | DMSO : 250 mg/mL (424.33 mM; Need ultrasonic) |
| form | Powder |
| pka | 13.82±0.20(Predicted) |
| color | White to off-white |
Description and Uses
Melanocortin 4 receptors play important roles in the regulation of energy homeostasis, eating behavior and sexual functions (1). (3R)-N-[(1R)-1-[(4-Chlorophenyl)methyl]-2-[4-cyclohexyl-4-(1H-1,2,4-triazol-1-ylmethyl)-1-piperidinyl]-2-oxoethyl]-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide is a potent and selective melanocortin 4 receptor agonist (2,3). It inhibits parasympathetic preganglionic neurons in the brainstem and regulates sympathetic and parasympathetic preganglionic neurons.
Safety
| Symbol(GHS) |  GHS07 |
| Signal word | Warning |
| Hazard statements | H302-H315-H319-H335 |
| Precautionary statements | P261-P305+P351+P338 |
