A7810012
Trelagliptin , ≥98% , 865759-25-7
CAS NO.:865759-25-7
Empirical Formula: C18H20FN5O2
Molecular Weight: 357.38
MDL number:
EINECS: 1592732-453-0
Pack Size | Price | Stock | Quantity |
5MG | RMB557.60 | In Stock |
|
10MG | RMB790.40 | In Stock |
|
25mg | RMB1759.20 | In Stock |
|
50MG | RMB3439.20 | In Stock |
|
100mg | RMB5583.20 | In Stock |
|
others | Enquire |
Update time: 2022-07-08
PRODUCT Properties
Boiling point: | 519.0±60.0 °C(Predicted) |
Density | 1.38±0.1 g/cm3(Predicted) |
storage temp. | Store at -20°C |
solubility | ≥11.6 mg/mL in DMSO; ≥3.68 mg/mL in EtOH with gentle warming and ultrasonic; ≥93.8 mg/mL in H2O |
form | solid |
pka | 9.88±0.20(Predicted) |
color | White to off-white |
InChI | InChI=1S/C18H20FN5O2/c1-22-17(25)8-16(23-6-2-3-15(21)11-23)24(18(22)26)10-13-7-14(19)5-4-12(13)9-20/h4-5,7-8,15H,2-3,6,10-11,21H2,1H3/t15-/m1/s1 |
InChIKey | IWYJYHUNXVAVAA-OAHLLOKOSA-N |
SMILES | C(#N)C1=CC=C(F)C=C1CN1C(=O)N(C)C(=O)C=C1N1CCC[C@@H](N)C1 |
Description and Uses
Trelagliptin is a highly selective, long-acting dipeptidyl peptidase IV (DPP-4) inhibitor. This inhibitor provides sustained reduction of plasma DPP-4 activity and lowering of blood glucose in animal models of diabetes.
Safety
Symbol(GHS) | GHS07 |
Signal word | Warning |
Hazard statements | H302-H315-H319-H335 |
Precautionary statements | P261-P280-P301+P312-P302+P352-P305+P351+P338 |