LN4514149
Efaroxanhydrochloride , ≥98% , 89197-00-2
Synonym(s):
2-Ethyl-2-(imidazolin-2-yl)-2,3-dihydrobenzofuran hydrochloride;RX 821037A
| Pack Size | Price | Stock | Quantity |
| 10mg | RMB488.00 | In Stock |
|
| 50mg | RMB1160.00 | In Stock |
|
| others | Enquire |
Update time: 2022-07-08
PRODUCT Properties
| storage temp. | Store at RT |
| solubility | H2O: 300 mg/mL |
| form | solid |
| color | White |
| Water Solubility | Soluble to 100 mM in water |
| Stability: | Stable for 1 year from date of purchase as supplied. Solutions in distilled water may be stored at -20° for up to 1 month. |
Description and Uses
Efaroxan HCl (89197-00-2) is a selective α2-adrenergic receptor antagonist1 (selectivity ratio of α2/α1 = 724)4 and imidazoline receptor antagonist2. Induces release of insulin in the rat insulinoma cell line RIN-5AH by interaction with ATP-sensitive potassium channels independently from imidazoline I1 or I2 receptors.3 Efaroxan HCl increases resting plasma insulin levels and markedly potentiates the rise in insulin levels produced by adrenaline in the rat.4
Efaroxan Hydrochloride is a potent α2-AR adrenoceptor antagonist.
